Peptide

Tesofensine

Triple reuptake weight loss

A triple monoamine reuptake inhibitor originally developed for Parkinson's that showed remarkable weight loss effects. Affects dopamine, serotonin, and norepinephrine.

Mechanisms

  • Triple reuptake inhibition
  • Appetite suppression
  • Metabolic enhancement

Dosing

Typical dose

0.25–0.5mg

Timing

Oral daily dosing. Significant weight loss potential.